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 Übersetzung für 'CB1' von Englisch nach Deutsch
biochem.
cannabinoid receptor type 1 <CNR1, CB1, CANN6, CB-R, CB1A, CB1K5, CB1R, CNR>
Cannabinoid-Rezeptor 1 {m} <CNR1, CB1, CNR, CB-R, CB1A, CANN6, CB1K5>
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  • Cannabinoid-Rezeptor 1 {m} <CNR1, CB1, CNR, CB-R, CB1A, CANN6, CB1K5> = cannabinoid receptor type 1 <CNR1, CB1, CANN6, CB-R, CB1A, CB1K5, CB1R, CNR>
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Anwendungsbeispiele Englisch
  • AM-919 is somewhat less potent than HU-210 itself, but is still a potent agonist at both CB1 and CB2 with moderate selectivity for CB1, with a Ki of 2.2 nM at CB1 and 3.4 nM at CB2.
  • AMG-1 is a potent agonist at both CB1 and CB2 with moderate selectivity for CB1, with a Ki of 0.6 nM at CB1 vs 3.1 nM at CB2.
  • AMG-36 is a potent agonist at both CB1 and CB2 with moderate selectivity for CB1, with a Ki of 0.45 nM at CB1 vs 1.92 nM at CB2.
  • NESS-0327 is a drug used in scientific research which acts as an extremely potent and selective antagonist of the cannabinoid receptor CB1.
  • JWH-018 is a full agonist of both the CB1 and CB2 cannabinoid receptors, with a reported binding affinity of 9.00 ± 5.00 nM at CB1 and 2.94 ± 2.65 nM at CB2.

  • CB1 selective antagonists are used for weight reduction and smoking cessation (see Rimonabant).
  • THCV is a cannabinoid receptor type 1 antagonist or, at higher doses, a CB1 receptor agonist and cannabinoid receptor type 2 partial agonist.
  • It has high affinity and efficacy at both the CB1 and CB2 cannabinoid receptors, with a Ki of 0.4nM at both CB1 and CB2, and an EC50 of ~0.06nM at CB1 and 0.2nM at CB2, making it one of the most potent cannabinoid agonists identified to date.
  • JWH-146 (1-heptyl-5-phenyl-1H-pyrrol-3-yl)-1-naphthalenyl-methanone) is a synthetic cannabinoid from the naphthoylpyrrole family which acts as an agonist of the CB1 (Ki = 21 ± 2nM) and CB2 (Ki = 62 ± 5nM) receptors, with a moderate (~2.9x) selectivity for the CB1 receptor over the CB2 receptor.
  • -naphthalen-1-ylmethanone) is a synthetic cannabinoid from the naphthoylpyrrole family which acts as an agonist of the CB1 (Ki = 53 ± 2nM) and CB2 (Ki = 23 ± 1nM) receptors, binding ~2.3 times stronger to the CB2 receptor than to the CB1 receptor.

  • -naphthalen-1-ylmethanone) is a synthetic cannabinoid from the naphthoylpyrrole family which acts as an agonist of the CB1 (Ki = 16 ± 1nM) and CB2 (Ki = 9.1 ± 0.7nM) receptors, binding ~1.76 times stronger to the CB2 receptor than to the CB1 receptor.
  • -naphthalen-1-ylmethanone) is a synthetic cannabinoid from the naphthoylpyrrole family which acts as an agonist of the CB1 (Ki = 42 ± 1nM) and CB2 (Ki = 64 ± 2nM) receptors, binding ~1.5 times stronger to the CB1 receptor than the CB2 receptor.
  • PipISB is a drug used in scientific research which acts as a potent and selective inverse agonist of the cannabinoid receptor CB1.
  • JWH-047 is a selective cannabinoid ligand that binds to both CB1 and CB2. It has a bindining affinity of Ki = 0.9 nM for the CB2 subtype, and more than 65 times selectivity over the CB1.
  • 3 nM and human CB1 receptors at Ki = 162.4 +/- 7.6 nM and functions as an agonist in human cannabinoid receptors but functions differently in rat cannabinoid receptors binding to rat cannabinoid CB2 receptors at Ki = 16.3 +/- 2.1 and CB1 receptors at Ki = 1130 +/- 574 nM binding to rat CB1 receptors 6.9x weaker than human CB1 receptors but increased binding for CB2.

  • Harrison founded CB1 Capital in 2017. CB1 Capital is a long-short healthcare hedge fund that intends to invest in the universe of stocks and industries that focus on cannabinoid-based solutions and other cannabis-based bio-pharmaceutical applications and therapies.
  • Org 27569 is a drug which acts as a potent and selective negative allosteric modulator of the cannabinoid CB1 receptor.
  • JWH-210 is an analgesic chemical from the naphthoylindole family, which acts as a potent cannabinoid agonist at both the CB1 and CB2 receptors, with Ki values of 0.46 nM at CB1 and 0.69 nM at CB2.
  • AM-694 (1-(5-fluoropentyl)-3-(2-iodobenzoyl)indole) is a designer drug that acts as a potent and selective agonist for the cannabinoid receptor CB1.
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Enthält Übersetzungen von der TU Chemnitz sowie aus Mr Honey's Business Dictionary (nur Englisch/Deutsch).
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